Pharmacology · single question

What is the mechanism of action of carvedilol?

  1. Beta-blockade (reduces cardiac workload; also alpha-1 blockade)
  2. Calcium-channel blockade
  3. ACE inhibition
  4. Direct vasodilation via nitric oxide
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Correct answer: A. Beta-blockade (reduces cardiac workload; also alpha-1 blockade)

  • A. Correct. Carvedilol is a non-selective beta-blocker with alpha-1 blocking activity; it lowers heart rate/contractility, reducing myocardial workload.
  • B. CCBs (e.g., amlodipine) act on calcium channels — a different class.
  • C. ACE inhibitors (e.g., lisinopril) block angiotensin conversion.
  • D. Direct NO vasodilation describes nitrates/hydralazine, not carvedilol.

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