Pharmacology · single question

What is the mechanism of action of prazosin?

  1. Alpha-1 adrenergic receptor antagonist
  2. Beta-1 blocker
  3. ACE inhibitor
  4. Calcium channel blocker
Show answer and explanation

Correct answer: A. Alpha-1 adrenergic receptor antagonist

  • A. Correct. Prazosin blocks alpha-1 receptors causing vasodilation; side effects include dizziness and orthostatic hypotension.
  • B. Beta-1 blockade describes atenolol/metoprolol.
  • C. ACE inhibition is a separate mechanism.
  • D. Prazosin does not act on calcium channels.

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