Pharmacology · single question

Mechanism of action of albuterol?

  1. Beta-2 adrenergic agonist
  2. Beta-1 agonist
  3. Anticholinergic
  4. Beta blocker
Show answer and explanation

Correct answer: A. Beta-2 adrenergic agonist

  • A. Correct. Albuterol is a selective beta-2 agonist that relaxes bronchial smooth muscle (bronchodilation) in asthma.
  • B. Incorrect. Beta-1 stimulation acts on the heart, not the primary bronchodilatory target.
  • C. Incorrect. Anticholinergics (e.g., ipratropium) bronchodilate by a different mechanism.
  • D. Incorrect. A beta blocker would WORSEN bronchospasm, the opposite of albuterol.

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