Pharmacology · single question

Lisinopril lowers blood pressure by:

  1. Inhibiting angiotensin-converting enzyme (blocking angiotensin I → angiotensin II)
  2. Blocking angiotensin II receptors
  3. Blocking beta-adrenergic receptors
  4. Blocking L-type calcium channels
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Correct answer: A. Inhibiting angiotensin-converting enzyme (blocking angiotensin I → angiotensin II)

  • A. Correct. Lisinopril is an ACE inhibitor: it blocks conversion of angiotensin I to angiotensin II, reducing vasoconstriction and aldosterone (a dry cough from bradykinin is a classic side effect).
  • B. ARBs (e.g., losartan) block the angiotensin II receptor — a different class.
  • C. Beta-blockers (e.g., metoprolol) act on adrenergic receptors.
  • D. Calcium-channel blockers (e.g., amlodipine) act on calcium channels.

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