Pharmacology · single question

What is the mechanism of action of albuterol?

  1. Beta-2 adrenergic agonist → bronchodilation
  2. Beta-2 adrenergic antagonist → bronchoconstriction
  3. Alpha-1 agonist → vasoconstriction
  4. Muscarinic antagonist → bronchodilation
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Correct answer: A. Beta-2 adrenergic agonist → bronchodilation

Albuterol is a selective Beta-2 adrenergic agonist (SABA — short-acting beta agonist). It stimulates β2-receptors on bronchial smooth muscle → increases cAMP → smooth muscle relaxation → bronchodilation. It's used for acute bronchospasm in asthma. A beta-2 ANTAgonist would cause bronchoconstriction. Ipratropium is the muscarinic antagonist bronchodilator.

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