Pharmacology · single question

Dexamethasone is best classified pharmacologically as a:

  1. Glucocorticoid antagonist
  2. Glucocorticoid agonist
  3. Mineralocorticoid agonist
  4. Mineralocorticoid antagonist
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Correct answer: B. Glucocorticoid agonist

  • A. It activates, rather than blocks, the glucocorticoid receptor.
  • B. Correct. Dexamethasone is a potent synthetic glucocorticoid receptor AGONIST with minimal mineralocorticoid activity.
  • C. It is not primarily a mineralocorticoid agonist (negligible mineralocorticoid effect).
  • D. Spironolactone is a mineralocorticoid antagonist; dexamethasone is not.

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