Pharmacology · single question

A patient needs a drug causing short-term anterograde amnesia (a diazepam-family drug). Which property is responsible?

  1. Serotonin reuptake inhibition
  2. GABA-A receptor potentiation (positive allosteric modulation)
  3. Dopamine D2 antagonism
  4. Muscarinic antagonism
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Correct answer: B. GABA-A receptor potentiation (positive allosteric modulation)

GABA-A receptor potentiation Benzodiazepines (midazolam is the classic choice for dental sedation because of its marked amnestic effect) cause anterograde amnesia by potentiating GABA-A-mediated inhibition in limbic structures. This is why midazolam is used for conscious sedation.

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